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The last 5 uploaded publications
Structure-based design of novel 2,4,5-trisubstituted pyrimidine derivatives as potent HIV-1 NNRTIs by exploiting the tolerant regions in NNTRIs binding pocket
Zhenzhen Zhou, Minghui Xie, Zongji Zhuo, Yalin Wang, Fabao Zhao, Sining Tao, Zhening Liang, De Clercq Erik, Christophe Pannecouque, Shujing Xu, Dongwei Kang, Xinyong Liu (2025). Structure-based design of novel 2,4,5-trisubstituted pyrimidine derivatives as potent HIV-1 NNRTIs by exploiting the tolerant regions in NNTRIs binding pocket. , 289, DOI: https://doi.org/10.1016/j.ejmech.2025.117464.
Article80 days agoStructure-Based Design of Novel 2,4,5-Trisubstituted Pyrimidine Derivatives as Potent Hiv-1 Nnrtis by Exploiting the Tolerant Regions in Nntris Binding Pocket
Zhenzhen Zhou, Minghui Xie, Zongji Zhuo, Sining Tao, Zhening Liang, De Clercq Erik, Christophe Pannecouque, Peng Zhan, Dongwei Kang, Xinyong Liu (2025). Structure-Based Design of Novel 2,4,5-Trisubstituted Pyrimidine Derivatives as Potent Hiv-1 Nnrtis by Exploiting the Tolerant Regions in Nntris Binding Pocket. , DOI: https://doi.org/10.2139/ssrn.5073546.
Preprint80 days agoDiscovery of low‐molecular‐weight phenylalanine derivatives as novel HIV capsid modulators with improved antiretroviral activity and metabolic stability
Xiangyi Jiang, Zhen Gao, Prem P. Sharma, Sumit Kumar, Brijesh Rathi, Xiangkai Ji, Jiaojiao Dai, Minghui Xie, Guanyu Dong, Shujing Xu, De Clercq Erik, Christophe Pannecouque, Alexej Dick, Peng Zhan, Xinyong Liu (2024). Discovery of low‐molecular‐weight phenylalanine derivatives as novel HIV capsid modulators with improved antiretroviral activity and metabolic stability. , 96(4), DOI: https://doi.org/10.1002/jmv.29594.
Article80 days agoDesign and optimization of piperidine-substituted thiophene[3,2-d]pyrimidine-based HIV-1 NNRTIs with improved drug resistance and pharmacokinetic profiles
Yanying Sun, Zhenzhen Zhou, Zhongling Shi, Fabao Zhao, Minghui Xie, Zongji Zhuo, De Clercq Erik, Christophe Pannecouque, Dongwei Kang, Peng Zhan, Xinyong Liu (2024). Design and optimization of piperidine-substituted thiophene[3,2-d]pyrimidine-based HIV-1 NNRTIs with improved drug resistance and pharmacokinetic profiles. , 14(7), DOI: https://doi.org/10.1016/j.apsb.2024.03.021.
Article80 days agoStructure‐based design of diarylpyrimidines and triarylpyrimidines as potent HIV‐1 NNRTIs with improved metabolic stability and drug resistance profiles
Minghui Xie, Zhao Wang, Fabao Zhao, Li Ye, Zongji Zhuo, Xin Li, De Clercq Erik, Christophe Pannecouque, Peng Zhan, Xinyong Liu, Dongwei Kang (2024). Structure‐based design of diarylpyrimidines and triarylpyrimidines as potent HIV‐1 NNRTIs with improved metabolic stability and drug resistance profiles. , 96(3), DOI: https://doi.org/10.1002/jmv.29502.
Article80 days ago