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The last 5 uploaded publications
Crystallographic and Receptor Binding Characterization of <i>Plasmodium falciparum</i> Macrophage Migration Inhibitory Factor Complexed to Two Potent Inhibitors
Georgios Pantouris, Deepa Rajasekaran, Alvaro Baeza Garcia, Victor G. Ruiz, Lin Leng, William L. Jorgensen, Richard Bucala, Elias Lolis (2014). Crystallographic and Receptor Binding Characterization of <i>Plasmodium falciparum</i> Macrophage Migration Inhibitory Factor Complexed to Two Potent Inhibitors. Journal of Medicinal Chemistry, 57(20), pp. 8652-8656, DOI: 10.1021/jm501168q.
Article360 days agoNovel allosteric covalent inhibitors of bifunctional Cryptosporidium hominis TS-DHFR from parasitic protozoa identified by virtual screening
Victor G. Ruiz, Daniel J. Czyzyk, Margarita Valhondo, William L. Jorgensen, Karen S. Anderson (2019). Novel allosteric covalent inhibitors of bifunctional Cryptosporidium hominis TS-DHFR from parasitic protozoa identified by virtual screening. Bioorganic & Medicinal Chemistry Letters, 29(11), pp. 1413-1418, DOI: 10.1016/j.bmcl.2019.03.022.
Article360 days agoTargeting the TS dimer interface in bifunctional Cryptosporidium hominis TS-DHFR from parasitic protozoa: Virtual screening identifies novel TS allosteric inhibitors
Victor G. Ruiz, Daniel J. Czyzyk, Vidya P. Kumar, William L. Jorgensen, Karen S. Anderson (2020). Targeting the TS dimer interface in bifunctional Cryptosporidium hominis TS-DHFR from parasitic protozoa: Virtual screening identifies novel TS allosteric inhibitors. Bioorganic & Medicinal Chemistry Letters, 30(16), pp. 127292-127292, DOI: 10.1016/j.bmcl.2020.127292.
Article360 days agoNovel allosteric covalent inhibitors of bifunctional Cryptosporidium hominis TS-DHFR from parasitic protozoa identified by virtual screening
Victor G. Ruiz, Daniel J. Czyzyk, Margarita Valhondo, William L. Jorgensen, Karen S. Anderson (2019). Novel allosteric covalent inhibitors of bifunctional Cryptosporidium hominis TS-DHFR from parasitic protozoa identified by virtual screening. Bioorganic & Medicinal Chemistry Letters, 29(11), pp. 1413-1418, DOI: 10.1016/j.bmcl.2019.03.022.
Article358 days ago