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The last 5 uploaded publications
Design, synthesis and structure-activity relationships of novel HIV capsid inhibitors with potent antiviral activities
Dazhou Shi, Shujing Xu, Lin Sun, Prem P. Sharma, Brijesh Rathi, Mei Wang, Linan Wu, Xiangyi Jiang, De Clercq Erik, Christophe Pannecouque, Xinyong Liu, Alexej Dick, Shujing Xu (2025). Design, synthesis and structure-activity relationships of novel HIV capsid inhibitors with potent antiviral activities. , 295, DOI: https://doi.org/10.1016/j.ejmech.2025.117784.
Article46 days agoDesign, Synthesis and Structure-Activity Relationships of Novel HIV Capsid Inhibitors with Potent Antiviral Activities
Dazhou Shi, Shujing Xu, Lin Sun, Prem P. Sharma, Brijesh Rathi, Mei Wang, Linan Wu, Xiangyi Jiang, De Clercq Erik, Christophe Pannecouque, Xinyong Liu, Alexej Dick, Peng Zhan (2025). Design, Synthesis and Structure-Activity Relationships of Novel HIV Capsid Inhibitors with Potent Antiviral Activities. , DOI: https://doi.org/10.2139/ssrn.5200966.
Preprint46 days agoDiscovery of low‐molecular‐weight phenylalanine derivatives as novel HIV capsid modulators with improved antiretroviral activity and metabolic stability
Xiangyi Jiang, Zhen Gao, Prem P. Sharma, Sumit Kumar, Brijesh Rathi, Xiangkai Ji, Jiaojiao Dai, Minghui Xie, Guanyu Dong, Shujing Xu, De Clercq Erik, Christophe Pannecouque, Alexej Dick, Peng Zhan, Xinyong Liu (2024). Discovery of low‐molecular‐weight phenylalanine derivatives as novel HIV capsid modulators with improved antiretroviral activity and metabolic stability. , 96(4), DOI: https://doi.org/10.1002/jmv.29594.
Article46 days agoDesign, Synthesis and Structure—Activity Relationships of Phenylalanine-Containing Peptidomimetics as Novel HIV-1 Capsid Binders Based on Ugi Four-Component Reaction
Xiangkai Ji, Jing Li, Prem P. Sharma, Xiangyi Jiang, Brijesh Rathi, Zhen Gao, Lide Hu, Dongwei Kang, De Clercq Erik, Simon Cocklin, Chuanfeng Liu, Christophe Pannecouque, Alexej Dick, Xinyong Liu, Peng Zhan (2022). Design, Synthesis and Structure—Activity Relationships of Phenylalanine-Containing Peptidomimetics as Novel HIV-1 Capsid Binders Based on Ugi Four-Component Reaction. , 27(18), DOI: https://doi.org/10.3390/molecules27185995.
Article46 days agoBoronic acid-containing diarylpyrimidine derivatives as novel HIV-1 NNRTIs: Design, synthesis and biological evaluation
Da Feng, Fenju Wei, Yanying Sun, Prem P. Sharma, Tao Zhang, Hao Lin, Brijesh Rathi, De Clercq Erik, Christophe Pannecouque, Dongwei Kang, Peng Zhan, Xinyong Liu (2021). Boronic acid-containing diarylpyrimidine derivatives as novel HIV-1 NNRTIs: Design, synthesis and biological evaluation. , 32(12), DOI: https://doi.org/10.1016/j.cclet.2021.02.033.
Article46 days ago