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The last 5 uploaded publications
A Fluorescence Polarization Assay for Binding to Macrophage Migration Inhibitory Factor and Crystal Structures for Complexes of Two Potent Inhibitors
José A. Cisneros, Michael J. Robertson, Margarita Valhondo, William L. Jorgensen (2016). A Fluorescence Polarization Assay for Binding to Macrophage Migration Inhibitory Factor and Crystal Structures for Complexes of Two Potent Inhibitors. Journal of the American Chemical Society, 138(27), pp. 8630-8638, DOI: 10.1021/jacs.6b04910.
Article361 days agoIrregularities in enzyme assays: The case of macrophage migration inhibitory factor
José A. Cisneros, Michael J. Robertson, Margarita Valhondo, William L. Jorgensen (2016). Irregularities in enzyme assays: The case of macrophage migration inhibitory factor. Bioorganic & Medicinal Chemistry Letters, 26(12), pp. 2764-2767, DOI: 10.1016/j.bmcl.2016.04.074.
Article361 days agoCovalent Inhibition of Wild-Type HIV-1 Reverse Transcriptase Using a Fluorosulfate Warhead
Joseph A. Ippolito, Haichan Niu, Nicole Bertoletti, Zachary J. Carter, Shengyan Jin, Krasimir A. Spasov, José A. Cisneros, Margarita Valhondo, Kara J. Cutrona, Karen S. Anderson, William L. Jorgensen (2021). Covalent Inhibition of Wild-Type HIV-1 Reverse Transcriptase Using a Fluorosulfate Warhead. ACS Medicinal Chemistry Letters, 12(2), pp. 249-255, DOI: 10.1021/acsmedchemlett.0c00612.
Article361 days agoNovel allosteric covalent inhibitors of bifunctional Cryptosporidium hominis TS-DHFR from parasitic protozoa identified by virtual screening
Victor G. Ruiz, Daniel J. Czyzyk, Margarita Valhondo, William L. Jorgensen, Karen S. Anderson (2019). Novel allosteric covalent inhibitors of bifunctional Cryptosporidium hominis TS-DHFR from parasitic protozoa identified by virtual screening. Bioorganic & Medicinal Chemistry Letters, 29(11), pp. 1413-1418, DOI: 10.1016/j.bmcl.2019.03.022.
Article361 days agoStructure activity relationship towards design of cryptosporidium specific thymidylate synthase inhibitors
Daniel J. Czyzyk, Margarita Valhondo, Luca Deiana, Julian Tirado‐Rives, William L. Jorgensen, Karen S. Anderson (2019). Structure activity relationship towards design of cryptosporidium specific thymidylate synthase inhibitors. European Journal of Medicinal Chemistry, 183, pp. 111673-111673, DOI: 10.1016/j.ejmech.2019.111673.
Article361 days ago