Simple heteroaryl modifications in the 4,5-diarylisoxazol-3-carboxylic acid scaffold favorably modulates the activity as dual mPGES-1/5-LO inhibitors with in vivo efficacy
Tuğba Gürses, Abdurrahman Olğaç, Ulrike Garscha, Tuğçe Gür Maz, Nur Banu Bal, Orhan Uludağ, Burcu Çalışkan, Ulrich Sigmar Schubert, Oliver Werz, Erden Banoğlu (2021). Simple heteroaryl modifications in the 4,5-diarylisoxazol-3-carboxylic acid scaffold favorably modulates the activity as dual mPGES-1/5-LO inhibitors with in vivo efficacy. , 112, DOI: https://doi.org/10.1016/j.bioorg.2021.104861.