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The last 5 uploaded publications
Optimization of novel di-substituted cyclohexylbenzamide derivatives as potent 11β-HSD1 inhibitors
Dustin L. McMinn, Yosup Rew, Athena Sudom, Seb Caille, Michael DeGraffenreid, Xiaodong He, Randall W. Hungate, Ben Jiang, Juan C. Jaén, Lisa D. Julian, Jacob A. Kaizerman, Perry M. Novak, Daqing Sun, Hua Tu, Stefania Ursu, Nigel P.C. Walker, Xuelei Yan, Qiuping Ye, Zhong Lin Wang, Jay P. Powers (2009). Optimization of novel di-substituted cyclohexylbenzamide derivatives as potent 11β-HSD1 inhibitors. , 19(5), DOI: https://doi.org/10.1016/j.bmcl.2009.01.026.
Article266 days agoDiscovery and optimization of piperidyl benzamide derivatives as a novel class of 11β-HSD1 inhibitors
Yosup Rew, Dustin L. McMinn, Zhong Lin Wang, Xiaodong He, Randall W. Hungate, Juan C. Jaén, Athena Sudom, Daqing Sun, Hua Tu, Stefania Ursu, Elisia Villemure, Nigel P.C. Walker, Xuelei Yan, Qiuping Ye, Jay P. Powers (2009). Discovery and optimization of piperidyl benzamide derivatives as a novel class of 11β-HSD1 inhibitors. , 19(6), DOI: https://doi.org/10.1016/j.bmcl.2009.01.058.
Article266 days agoDiscovery of Novel, Potent Benzamide Inhibitors of 11β-Hydroxysteroid Dehydrogenase Type 1 (11β-HSD1) Exhibiting Oral Activity in an Enzyme Inhibition ex Vivo Model<sup>▽</sup>
Lisa D. Julian, Zhong Lin Wang, Tracy Bostick, Seb Caille, Rebekah Choi, Michael DeGraffenreid, Yongmei Di, Xiaodong He, Randall W. Hungate, Juan C. Jaén, Jinsong Liu, Mario Monshouwer, Dustin L. McMinn, Yosup Rew, Athena Sudom, Daqing Sun, Hua Tu, Stefania Ursu, Nigel P.C. Walker, Xuelei Yan, Qiuping Ye, Jay P. Powers (2008). Discovery of Novel, Potent Benzamide Inhibitors of 11β-Hydroxysteroid Dehydrogenase Type 1 (11β-HSD1) Exhibiting Oral Activity in an Enzyme Inhibition ex Vivo Model<sup>▽</sup>. , 51(13), DOI: https://doi.org/10.1021/jm800310g.
Article266 days agoSynthesis and optimization of novel 4,4-disubstituted cyclohexylbenzamide derivatives as potent 11β-HSD1 inhibitors
Daqing Sun, Zhong Lin Wang, Seb Caille, Michael DeGraffenreid, Felix González-López de Turiso, Randall W. Hungate, Juan C. Jaén, Ben Jiang, Lisa D. Julian, Ron C. Kelly, Dustin L. McMinn, Jacob A. Kaizerman, Yosup Rew, Athena Sudom, Hua Tu, Stefania Ursu, Nigel P.C. Walker, Maren Gulsrud Willcockson, Xuelei Yan, Qiuping Ye, Jay P. Powers (2010). Synthesis and optimization of novel 4,4-disubstituted cyclohexylbenzamide derivatives as potent 11β-HSD1 inhibitors. , 21(1), DOI: https://doi.org/10.1016/j.bmcl.2010.10.129.
Article262 days ago