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Won-Gil Lee, Kathleen M. Frey, Ricardo Gallardo‐Macias, Krasimir A. Spasov, Albert H. Chan, Karen S. Anderson, William L. Jorgensen (2015). Discovery and crystallography of bicyclic arylaminoazines as potent inhibitors of HIV-1 reverse transcriptase. Bioorganic & Medicinal Chemistry Letters, 25(21), pp. 4824-4827, DOI: 10.1016/j.bmcl.2015.06.074.