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The last 5 uploaded publications
Design, synthesis, and biological evaluation of piperidinyl‐substituted [1,2,4]triazolo[1,5‐a]pyrimidine derivatives as potential anti‐HIV‐1 agents with reduced cytotoxicity
Boshi Huang, Dongwei Kang, Ye Tian, Dirk Daelemans, De Clercq Erik, Christophe Pannecouque, Peng Zhan, Xinyong Liu (2020). Design, synthesis, and biological evaluation of piperidinyl‐substituted [1,2,4]triazolo[1,5‐a]pyrimidine derivatives as potential anti‐HIV‐1 agents with reduced cytotoxicity. , 97(1), DOI: https://doi.org/10.1111/cbdd.13760.
Article36 days agoDiscovery of novel diarylpyrimidines as potent HIV NNRTIs via a structure-guided core-refining approach
Xiao Li, Wen‐Ming Chen, Ye Tian, Huiqing Liu, Peng Zhan, De Clercq Erik, Christophe Pannecouque, Jan Balzarini, Xinyong Liu (2014). Discovery of novel diarylpyrimidines as potent HIV NNRTIs via a structure-guided core-refining approach. , 80, DOI: https://doi.org/10.1016/j.ejmech.2014.04.036.
Article36 days agoDesign, Synthesis, and Biological Evaluation of Novel 3,5‐Disubstituted‐1,2,6‐Thiadiazine‐1,1‐Dione Derivatives as <scp>HIV</scp>‐1 <scp>NNRTI</scp>s
Ye Tian, Diwakar Rai, Peng Zhan, Christophe Pannecouque, Jan Balzarini, De Clercq Erik, Huiqing Liu, Xinyong Liu (2013). Design, Synthesis, and Biological Evaluation of Novel 3,5‐Disubstituted‐1,2,6‐Thiadiazine‐1,1‐Dione Derivatives as <scp>HIV</scp>‐1 <scp>NNRTI</scp>s. , 82(4), DOI: https://doi.org/10.1111/cbdd.12160.
Article36 days agoDiscovery of Thiophene[3,2-<i>d</i>]pyrimidine Derivatives as Potent HIV-1 NNRTIs Targeting the Tolerant Region I of NNIBP
Dongwei Kang, Xiao Ding, Gaochan Wu, Zhipeng Huo, Zhongxia Zhou, Tong Zhao, Da Feng, Zhao Wang, Ye Tian, Dirk Daelemans, De Clercq Erik, Christophe Pannecouque, Peng Zhan, Xinyong Liu (2017). Discovery of Thiophene[3,2-<i>d</i>]pyrimidine Derivatives as Potent HIV-1 NNRTIs Targeting the Tolerant Region I of NNIBP. , 8(11), DOI: https://doi.org/10.1021/acsmedchemlett.7b00361.
Article36 days agoStructure-Based Optimization of Thiophene[3,2-<i>d</i>]pyrimidine Derivatives as Potent HIV-1 Non-nucleoside Reverse Transcriptase Inhibitors with Improved Potency against Resistance-Associated Variants
Dongwei Kang, Zengjun Fang, Boshi Huang, Xueyi Lu, Heng Zhang, Haoran Xu, Zhipeng Huo, Zhongxia Zhou, Yu Zhao, Qing Meng, Gaochan Wu, Xiao Ding, Ye Tian, Dirk Daelemans, De Clercq Erik, Christophe Pannecouque, Peng Zhan, Xinyong Liu (2017). Structure-Based Optimization of Thiophene[3,2-<i>d</i>]pyrimidine Derivatives as Potent HIV-1 Non-nucleoside Reverse Transcriptase Inhibitors with Improved Potency against Resistance-Associated Variants. , 60(10), DOI: https://doi.org/10.1021/acs.jmedchem.7b00332.
Article36 days ago