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The last 5 uploaded publications
Engineering diaminotriazole ligands into ATP-mimetics for selective targeting of the Janus kinase 2 (JAK2) pseudokinase domain (JH2)
Maria-Elena Liosi, Stefan Krimmer, Ana S. Newton, Thomas L. Dawson, David A. Puleo, Kara J. Cutrona, Yoshihisa Suzuki, Sean Henry, Joseph Schlessinger, William L. Jorgensen (2021). Engineering diaminotriazole ligands into ATP-mimetics for selective targeting of the Janus kinase 2 (JAK2) pseudokinase domain (JH2). , DOI: 10.1021/scimeetings.1c00737.
Preprint380 days agoIdentification and Characterization of JAK2 Pseudokinase Domain Small Molecule Binders
D.E. Puleo, Kaury Kucera, Henrik M. Hammarén, Daniela Ungureanu, Ana S. Newton, Olli Silvennoinen, William L. Jorgensen, Joseph Schlessinger (2017). Identification and Characterization of JAK2 Pseudokinase Domain Small Molecule Binders. ACS Medicinal Chemistry Letters, 8(6), pp. 618-621, DOI: 10.1021/acsmedchemlett.7b00153.
Article360 days agoInsights on JAK2 Modulation by Potent, Selective, and Cell-Permeable Pseudokinase-Domain Ligands
Maria-Elena Liosi, Joseph A. Ippolito, Sean P. Henry, S.G. Krimmer, Ana S. Newton, Kara J. Cutrona, Rene A. Olivarez, Jyotidarsini Mohanty, Joseph Schlessinger, William L. Jorgensen (2022). Insights on JAK2 Modulation by Potent, Selective, and Cell-Permeable Pseudokinase-Domain Ligands. Journal of Medicinal Chemistry, 65(12), pp. 8380-8400, DOI: 10.1021/acs.jmedchem.2c00283.
Article360 days agoJAK2 JH2 Fluorescence Polarization Assay and Crystal Structures for Complexes with Three Small Molecules
Ana S. Newton, Luca Deiana, D.E. Puleo, José A. Cisneros, Kara J. Cutrona, Joseph Schlessinger, William L. Jorgensen (2017). JAK2 JH2 Fluorescence Polarization Assay and Crystal Structures for Complexes with Three Small Molecules. ACS Medicinal Chemistry Letters, 8(6), pp. 614-617, DOI: 10.1021/acsmedchemlett.7b00154.
Article360 days agoSelective Janus Kinase 2 (JAK2) Pseudokinase Ligands with a Diaminotriazole Core
Maria-Elena Liosi, S.G. Krimmer, Ana S. Newton, Thomas K. Dawson, D.E. Puleo, Kara J. Cutrona, Yoshihisa Suzuki, Joseph Schlessinger, William L. Jorgensen (2020). Selective Janus Kinase 2 (JAK2) Pseudokinase Ligands with a Diaminotriazole Core. Journal of Medicinal Chemistry, 63(10), pp. 5324-5340, DOI: 10.1021/acs.jmedchem.0c00192.
Article360 days ago