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The last 5 uploaded publications
Molecular Basis of Sphingosine Kinase 1 Substrate Recognition and Catalysis
Jinsong Liu, Jessica Dai, Songzhu An, Stephen Thibault, Nigel P.C. Walker, Zhong Lin Wang, Xiaoshan Min, Shou-Hua Xiao, Sheree Johnstone, William G. Romanow, David Meininger, Haoda Xu (2013). Molecular Basis of Sphingosine Kinase 1 Substrate Recognition and Catalysis. , 21(5), DOI: https://doi.org/10.1016/j.str.2013.02.025.
Article288 days agoDiscovery of Novel, Potent Benzamide Inhibitors of 11β-Hydroxysteroid Dehydrogenase Type 1 (11β-HSD1) Exhibiting Oral Activity in an Enzyme Inhibition ex Vivo Model<sup>▽</sup>
Lisa D. Julian, Zhong Lin Wang, Tracy Bostick, Seb Caille, Rebekah Choi, Michael DeGraffenreid, Yongmei Di, Xiaodong He, Randall W. Hungate, Juan C. Jaén, Jinsong Liu, Mario Monshouwer, Dustin L. McMinn, Yosup Rew, Athena Sudom, Daqing Sun, Hua Tu, Stefania Ursu, Nigel P.C. Walker, Xuelei Yan, Qiuping Ye, Jay P. Powers (2008). Discovery of Novel, Potent Benzamide Inhibitors of 11β-Hydroxysteroid Dehydrogenase Type 1 (11β-HSD1) Exhibiting Oral Activity in an Enzyme Inhibition ex Vivo Model<sup>▽</sup>. , 51(13), DOI: https://doi.org/10.1021/jm800310g.
Article288 days agoDistinctive molecular inhibition mechanisms for selective inhibitors of human 11β-hydroxysteroid dehydrogenase type 1
Hua Tu, Jay P. Powers, Jinsong Liu, Stefania Ursu, Athena Sudom, Xuelei Yan, Haoda Xu, David Meininger, Michael DeGraffenreid, Xiaodong He, Juan C. Jaén, Daqing Sun, Marc Labelle, Hiroshi Yamamoto, Bei Shan, Nigel P.C. Walker, Zhong Lin Wang (2008). Distinctive molecular inhibition mechanisms for selective inhibitors of human 11β-hydroxysteroid dehydrogenase type 1. , 16(19), DOI: https://doi.org/10.1016/j.bmc.2008.08.065.
Article288 days agoDiscovery of INT131: A selective PPARγ modulator that enhances insulin sensitivity
Joshua P. Taygerly, Lawrence R. McGee, Steven M. Rubenstein, Jonathan B. Houze, Timothy D. Cushing, Yang Li, Alykhan Motani, Jin-Long Chen, Walter Frankmoelle, Guosen Ye, Marc Learned, Juan C. Jaén, Shichang Miao, Pieter B.M.W.M. Timmermans, Martin Thoolen, Patricia M. Kearney, John A. Flygare, Holger Beckmann, Jennifer Weiszmann, Michelle Lindström, Nigel P.C. Walker, Jinsong Liu, Donna H.T. Biermann, Zhong Lin Wang, Atsushi Hagiwara, Tetsuya Iida, Hisateru Aramaki, Yuki Kitao, Hisashi Shinkai, Noboru Furukawa, Jun Nishiu, Motonao Nakamura (2012). Discovery of INT131: A selective PPARγ modulator that enhances insulin sensitivity. , 21(4), DOI: https://doi.org/10.1016/j.bmc.2012.11.058.
Article284 days agoThe synthesis and SAR of novel diarylsulfone 11β-HSD1 inhibitors
Xuelei Yan, Zhong Lin Wang, Athena Sudom, Mario Cardozo, Michael DeGraffenreid, Yongmei Di, Pingchen Fan, Xiaodong He, Juan C. Jaén, Marc Labelle, Jinsong Liu, Ji Ma, Dustin L. McMinn, Shichang Miao, Daqing Sun, Liang Tang, Hua Tu, Stefania Ursu, Nigel P.C. Walker, Qiuping Ye, Jay P. Powers (2010). The synthesis and SAR of novel diarylsulfone 11β-HSD1 inhibitors. , 20(23), DOI: https://doi.org/10.1016/j.bmcl.2010.09.097.
Article284 days ago