Design, synthesis, and biological evaluation of dual-site HIV-1 inhibitors simultaneously targeting the NNRTI binding pocket and an adjacent site with favorable resistance profiles
Xiangkai Ji, Xiangyi Jiang, X. T. Huang, Heng Gao, Zhen Gao, Ping Gao, De Clercq Erik, Christophe Pannecouque, Dongwei Kang, Peng Zhan, Xinyong Liu (2025). Design, synthesis, and biological evaluation of dual-site HIV-1 inhibitors simultaneously targeting the NNRTI binding pocket and an adjacent site with favorable resistance profiles. , 164, DOI: https://doi.org/10.1016/j.bioorg.2025.108924.