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The last 5 uploaded publications
Transcription factor Ascl2 promotes germinal center B cell responses by directly regulating AID transcription
Lin Sun, Xiaohong Zhao, Xindong Liu, Bo Zhong, Hong Tang, Wei Jin, Hans Clevers, Hui Wang, Xiaohu Wang, Chen Dong (2021). Transcription factor Ascl2 promotes germinal center B cell responses by directly regulating AID transcription. , 35(9), DOI: https://doi.org/10.1016/j.celrep.2021.109188.
Article123 days ago2,4,5-Trisubstituted Pyrimidines as Potent HIV-1 NNRTIs: Rational Design, Synthesis, Activity Evaluation, and Crystallographic Studies
Dongwei Kang, Francesc X. Ruiz, Yanying Sun, Da Feng, Lanlan Jing, Zhao Wang, Tao Zhang, Shenghua Gao, Lin Sun, De Clercq Erik, Christophe Pannecouque, Eddy Arnold, Peng Zhan, Xinyong Liu (2021). 2,4,5-Trisubstituted Pyrimidines as Potent HIV-1 NNRTIs: Rational Design, Synthesis, Activity Evaluation, and Crystallographic Studies. , 64(7), DOI: https://doi.org/10.1021/acs.jmedchem.1c00268.
Article35 days agoDesign, synthesis, and mechanism study of dimerized phenylalanine derivatives as novel HIV-1 capsid inhibitors
Xujie Zhang, Lin Sun, Megan E. Meuser, Waleed A. Zalloum, Shujing Xu, Tianguang Huang, Srinivasulu Cherukupalli, Xiangyi Jiang, Xiao Ding, Yucen Tao, Dongwei Kang, De Clercq Erik, Christophe Pannecouque, Alexej Dick, Simon Cocklin, Xinyong Liu, Peng Zhan (2021). Design, synthesis, and mechanism study of dimerized phenylalanine derivatives as novel HIV-1 capsid inhibitors. , 226, DOI: https://doi.org/10.1016/j.ejmech.2021.113848.
Article35 days agoDiscovery of potential dual-target prodrugs of HIV-1 reverse transcriptase and nucleocapsid protein 7
Songkai Sun, Boshi Huang, Zhuo Li, Zhao Wang, Lin Sun, Ping Gao, Dongwei Kang, Chin‐Ho Chen, Kuo‐Hsiung Lee, Dirk Daelemans, De Clercq Erik, Christophe Pannecouque, Peng Zhan, Xinyong Liu (2020). Discovery of potential dual-target prodrugs of HIV-1 reverse transcriptase and nucleocapsid protein 7. , 30(16), DOI: https://doi.org/10.1016/j.bmcl.2020.127287.
Article35 days agoDesign, Synthesis, and Mechanism Study of Benzenesulfonamide-Containing Phenylalanine Derivatives as Novel HIV-1 Capsid Inhibitors with Improved Antiviral Activities
Lin Sun, Alexej Dick, Megan E. Meuser, Tianguang Huang, Waleed A. Zalloum, Chin‐Ho Chen, Srinivasulu Cherukupalli, Shujing Xu, Xiao Ding, Ping Gao, Dongwei Kang, De Clercq Erik, Christophe Pannecouque, Simon Cocklin, Kuo‐Hsiung Lee, Xinyong Liu, Peng Zhan (2020). Design, Synthesis, and Mechanism Study of Benzenesulfonamide-Containing Phenylalanine Derivatives as Novel HIV-1 Capsid Inhibitors with Improved Antiviral Activities. , 63(9), DOI: https://doi.org/10.1021/acs.jmedchem.0c00015.
Article35 days ago